Compound | unP-IC50 (µM)1 | P-IC50 value (µM)2 | Ratio3 |
---|---|---|---|
Hit 1 | 10.0 | >100 | >10 |
Hit 2 | 14.0 | >60 | >4 |
Hit 3 | 27 | >100 | >4 |
Hit 4 | 19.0 | >60 | >3 |
Hit 5 | 11.0 | 59.0 | 5.4 |
Hit 6 | 15.0 | >100 | >7 |
Hit 7 | 2.5 | 2.5 | 1 |
Staurosporine | 0.028 | 0.057 | 2.0 |
SU11274 | 0.005 | 0.28 | 56.0 |